1. Signaling Pathways
  2. GPCR/G Protein
    Neuronal Signaling
  3. Dopamine Receptor
  4. Dopamine Receptor Inhibitors

Dopamine Receptor Inhibitors

Dopamine Receptor

D1 Receptor

D2 Receptor

D3 Receptor

D4 Receptor

D5 Receptor

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Dopamine Receptor Inhibitors, Agonists, Antagonists, Activators, Modulators, Controls & Ligands
Product Name Dopamine Receptor D1 Receptor D2 Receptor D3 Receptor D4 Receptor D5 Receptor Purity
Docarpamine  
D1 Receptor
       
SCH-23390 hydrochloride  
D1 Receptor, Ki: 0.2 nM
     
D5 Receptor, Ki: 0.3 nM
99.83%
Clozapine    
D2 Receptor, Ki: 75 nM (Antagonist)
      99.84%
Haloperidol    
D2 Receptor
      99.69%
Olanzapine
Dopamine Receptor
          99.96%
Risperidone    
D2 Receptor, Ki: 5.9 nM
      99.87%
Bromocriptine mesylate    
D2 Receptor
      99.98%
SKF 38393 hydrochloride  
D1 Receptor
        99.49%
WAY-100635        
D4 Receptor
  99.97%
Sulpiride    
D2 Receptor
D3 Receptor
    99.28%
Aripiprazole    
D2 Receptor
D3 Receptor
D4 Receptor
  99.93%
Brexpiprazole    
D2L Receptor, Ki: 0.3 nM
      99.80%
Penfluridol    
D2 Receptor
      99.93%
Raclopride  
D1 Receptor, Ki: 18000 nM
D2 Receptor, Ki: 1.8 nM
D3 Receptor, Ki: 3.5 nM
D4 Receptor, Ki: 2400 nM
  99.86%
Cabergoline    
D2 Receptor
D3 Receptor
    99.86%
SKF 81297  
D1 Receptor
        99.68%
Buspirone    
Dopamine D2 receptor
      99.86%
Tetrabenazine    
D2 Receptor, Ki: ~2.1 μM
      99.95%
Ritanserin    
D2 Receptor, IC50: 70 nM
      99.68%
SKF 81297 hydrobromide  
D1 Receptor
        99.88%
WAY-100635 maleate        
D4 Receptor
  99.57%
Nuciferine    
D2 Receptor, EC50: 64 nM
 
D4 Receptor, EC50: 2 μM
D5 Receptor, EC50: 2.6 μM
99.90%
Cariprazine    
D2 Receptor, Ki: 0.49 nM
D3 Receptor, Ki: 0.085 nM
    99.67%
Rotigotine  
D1 Receptor, Ki: 83 nM
D2 Receptor, Ki: 4-15 nM
D3 Receptor, Ki: 0.71 nM
D4 Receptor, Ki: 4-15 nM
D5 Receptor, Ki: 4-15 nM
99.98%
Ropinirole hydrochloride    
D2 Receptor, Ki: 29 nM
hD2 Receptor, pEC50: 7.4
hD3 Receptor, pEC50: 8.4
hD4.4 Receptor, pEC50: 6.8
  99.89%
Domperidone    
D2 Receptor
      99.87%
Sumanirole maleate    
D2 Receptor
      99.78%
N-Methyldopamine hydrochloride  
D1 Receptor
        99.12%
Ziprasidone    
Rat D2 Receptor, Ki: 4.8 nM
      99.31%
Perphenazine    
D2 Receptor, Ki: 0.56 nM
D3 Receptor, Ki: 0.43 nM
D4 Receptor, Ki: 28.5 nM
  99.81%
Paliperidone    
D2 Receptor
      99.43%
Prochlorperazine dimaleate    
D2 Receptor
      ≥98.0%
Cariprazine hydrochloride    
D2 Receptor, Ki: 0.49 nM
D3 Receptor, Ki: 0.085 nM
    99.88%
Rotigotine Hydrochloride  
D1 Receptor, Ki: 83 nM
D2 Receptor, Ki: 4-15 nM
D3 Receptor, Ki: 0.71 nM
D4 Receptor, Ki: 4-15 nM
D5 Receptor, Ki: 4-15 nM
99.45%
Amisulpride    
Human D2 Receptor, Ki: 2.8 nM
D3 Receptor, Ki: 3.2 nM
    99.77%
Pramipexole    
D2 Receptor, Ki: 3.9 nM
D3 Receptor, Ki: 0.5 nM
D4 Receptor, Ki: 1.3 nM
  99.88%
L-741626        
D4 Receptor
  99.0%
Pramipexole dihydrochloride    
D2 Receptor
D3 Receptor
D4 Receptor
  99.73%
SKF-82958 hydrobromide  
D1 Receptor
        99.53%
Lumateperone  
D1 Receptor
D2 Receptor
      99.83%
Lurasidone    
D2 Receptor, IC50: 1.68 nM
      99.36%
Benztropine mesylate    
Human D2 Receptor
      99.85%
Metoclopramide    
D2 Receptor, IC50: 483 nM
      99.98%
Loxapine succinate  
Human D1 Receptor
Human D2 Receptor
 
Human D4 Receptor
  98.84%
Eticlopride hydrochloride    
D2 Receptor, Ki: 0.09 nM
      99.45%
Rotundine  
D1 Receptor, IC50: 166 nM
D2 Receptor, IC50: 1400 nM
D3 Receptor, IC50: 3300 nM
    99.96%
Blonanserin  
D1 Receptor, Ki: 1070 nM
D2 Receptor, Ki: 0.142 nM
D3 Receptor, Ki: 0.494 nM
D4 Receptor, Ki: 150 nM
  99.91%
Flunarizine dihydrochloride    
D2 Receptor
      99.90%
Lisuride    
D2 Receptor
      99.85%
Dihydrexidine hydrochloride  
D1 Receptor, IC50: 10 nM
        98.89%
Pridopidine    
D2 Receptor
      99.85%
Flunarizine    
D2 Receptor
      99.79%
Ecopipam hydrochloride  
D1 Receptor, Ki: 1.2 nM
D2 Receptor, Ki: 980 nM
 
D4 Receptor, Ki: 5520 nM
D5 Receptor, Ki: 2.0 nM
99.46%
Loxapine  
Human D1 Receptor
Human D2 Receptor
 
Human D4 Receptor
  99.93%
SKF-83566  
D1 Receptor
     
D5 Receptor
99.86%
L-745870    
D2 Receptor, Ki: 960 nM
D3 Receptor, Ki: 2300 nM
Human D4 Receptor, Ki: 4.3 nM
  99.92%
Flupentixol dihydrochloride  
D1 Receptor
D2 Receptor
      99.73%
A68930 hydrochloride  
D1 Receptor
        98.71%
Bromperidol    
D2 Receptor
      99.83%
Chlorprothixene  
Human D1 Receptor, Ki: 18 nM
Human D2 Receptor, Ki: 2.96 nM
Human D3 Receptor, Ki: 4.56 nM
 
Human D5 Receptor, Ki: 9 nM
99.87%
UNC9994 hydrochloride  
D1 Receptor, Ki: 4000 nM
D2 Receptor, Ki: 79 nM
D3 Receptor, Ki: 17 nM
D4 Receptor, Ki: 138 nM
  99.50%
Promazine hydrochloride    
D2 Receptor
      99.87%
Iloperidone  
Rat D1 Receptor, Ki: 546 nM
Human D1 Receptor, Ki: 216 nM
Rat D2 Receptor, Ki: 54 nM
Human D3 Receptor, Ki: 7.1 nM
Human D4 Receptor, Ki: 25 nM
Human D5 Receptor, Ki: 319 nM
99.93%
Thiethylperazine    
D2 Receptor
      99.91%
UNC9995    
D2 Receptor
      99.93%
Talipexole dihydrochloride    
D2 Receptor
      99.80%
SB-277011 hydrochloride      
D3 Receptor, Ki: 10.7-11.2 nM
    99.59%
L-DOPA-2,5,6-d3      
D3 Receptor
    99.67%
MLS1547    
D2 Receptor
      99.94%
Piribedil    
D2 Receptor
D3 Receptor
    99.92%
Chlorprothixene hydrochloride  
Human D1 Receptor, Ki: 18 nM
Human D2 Receptor, Ki: 2.96 nM
Human D3 Receptor, Ki: 4.56 nM
 
Human D5 Receptor, Ki: 9 nM
99.91%
Itopride hydrochloride    
D2 Receptor
      99.84%
Paliperidone palmitate    
D2 Receptor
      99.93%
UCSF924        
D4 Receptor
  99.53%
Pramipexole dihydrochloride hydrate    
D2 Receptor, Ki: 3.9 nM
D3 Receptor, Ki: 0.5 nM
D4 Receptor, Ki: 1.3 nM
  98.0%
Asenapine  
D1 Receptor, pKi: 8.9
D2 Receptor, pKi: 8.9
D3 Receptor, pKi: 9.4
D4 Receptor, pKi: 9.0
  99.62%
Pericyazine    
D2 Receptor
      99.86%
PD-168077 maleate        
D4 Receptor
  99.60%
Dehydroaripiprazole    
D2 Receptor
D3 Receptor
    99.95%
Lumateperone tosylate  
D1 Receptor
D2 Receptor
      99.78%
Ansofaxine hydrochloride
Dopamine Receptor, IC50: 491 nM
          99.44%
L-745870 hydrochloride    
D2 Receptor, Ki: 960 nM
D3 Receptor, Ki: 2300 mM
Human D4 Receptor, Ki: 4.3 nM
  99.91%
Ziprasidone hydrochloride monohydrate    
Rat D2 Receptor, Ki: 4.8 nM
      98.11%
Lurasidone Hydrochloride    
D2 Receptor, IC50: 1.68 nM
      99.86%
Spiperone hydrochloride  
D1 Receptor, Ki: ~350 nM
D2 Receptor, Ki: 0.06 nM
D3 Receptor, Ki: 0.6 nM
D4 Receptor, Ki: 0.08 nM
D5 Receptor, Ki: ~3500 nM
99.10%
Zuclopenthixol    
D2 Receptor
      98.08%
(+)-PD 128907 hydrochloride    
D2 Receptor
D3 Receptor
    98.92%
Tetrabenazine Racemate    
D2 Receptor, Ki: ~2.1 μM
      99.89%
Metoclopramide hydrochloride hydrate    
D2 Receptor, IC50: 483 nM
      99.96%
SKF 83959  
D1 Receptor, Ki: 1.18 nM
D2 Receptor, Ki: 920 nM
D3 Receptor, Ki: 399 nM
 
D5 Receptor, Ki: 7.56 nM
98.30%
Ocaperidone    
D2 Receptor, Ki: 0.75 nM
      98.65%
D-Tetrahydropalmatine  
D1 Receptor
        99.84%
Amisulpride hydrochloride      
D3 Receptor
    99.79%
Oxypertine    
D2 Receptor, Ki: 30 nM
      99.84%
Xaliproden hydrochloride    
D2 Receptor
      98.40%
GR 103691      
D3 Receptor
    99.91%
Ecopipam  
D1 Receptor, Ki: 1.2 nM
D2 Receptor, Ki: 980 nM
 
D4 Receptor, Ki: 5520 nM
D5 Receptor, Ki: 2.0 nM
99.77%
Desmethyl cariprazine    
D2 Receptor, Ki: 0.49 nM
D3 Receptor, Ki: 0.085 nM
    98.08%
Tiapride hydrochloride    
D2 Receptor, IC50: 110-320 nM
D3 Receptor, IC50: 180 nM
    99.95%
Metopimazine    
D2 Receptor
      99.75%
GSK598809      
D3 Receptor
    99.73%
Sarizotan    
rD2 Receptor, IC50: 15.1 nM (rat)
hD2 Receptor, IC50: 17 nM
D3 Receptor, IC50: 6.8 nM (human)
hD4.2 Receptor, IC50: 2.4 nM
  98.23%
Neuromedin N    
D2 Receptor
      99.84%
Roxindole hydrochloride    
D2 Receptor
      99.48%
Propionylpromazine hydrochloride    
D2 Receptor
      99.71%
Fluphenazine decanoate    
D2 Receptor
      98.75%
Haloperidol hydrochloride    
D2 Receptor
      99.56%
Ziprasidone hydrochloride    
Rat D2 Receptor, Ki: 4.8 nM
      99.74%
ML417      
D3 Receptor, EC50: 38 nM
    99.39%
NGB 2904      
D3 Receptor, Ki: 1.4 nM
    99.76%
Bacopaside X  
D1 Receptor
        99.64%
Nemonapride    
D2 Receptor, Ki: 0.06 nM
      99.90%
Ropinirole    
D2 Receptor, Ki: 29 nM
hD2 Receptor, pEC50: 7.4
hD3 Receptor, pEC50: 8.4
hD4.4 Receptor, pEC50: 6.8
  99.42%
(Rac)-Tavapadon  
D1 Receptor
        99.49%
SKF 83822  
Rat D1 Receptor
        98.01%
Pipamperone    
D2 Receptor, pKi: 6.7
 
D4 Receptor, pKi: 8.0
  99.89%
Halopemide  
D1 Receptor
D2 Receptor
      99.65%
Melperone    
Human D2 Receptor, Kd: 180 nM
      99.84%
PG01037 dihydrochloride      
D3 Receptor, Ki: 0.7 nM
    99.35%
Naxagolide    
D2 Receptor
      99.81%
Didesmethyl cariprazine    
D2L Receptor, Ki: 1.41 nM
Human D3 Receptor, Ki: 0.056 nM
    99.63%
Brilaroxazine    
D2 Receptor
D3 Receptor
D4 Receptor
  98.82%
UNC9994    
D2 Receptor, Ki: 79 nM
D3 Receptor, Ki: 17 nM
D4 Receptor, Ki: 138 nM
  98.06%
CY 208-243  
D1 Receptor
        99.99%
Benztropine    
D2 Receptor
      98.12%
Thiethylperazine dimaleate    
D2 Receptor
      99.99%
Molindone hydrochloride    
D2 Receptor
   
D5 Receptor
99.78%
Acetophenazine dimaleate    
D2 Receptor
      99.90%
Dopamine D4 receptor antagonist-1        
hD4.2 Receptor, Ki: 9.0 nM
  98.59%
LE 300  
Human D1 Receptor, Ki: 1.9 nM
     
Human D5 Receptor, Ki: 7.5 nM
98.5%
Sonepiprazole    
rD2 Receptor, Ki: 5147 nM
 
rD4 Receptor, Ki: 3.6 nM
hD4.2 Receptor, Ki: 10.1 nM
  98.43%
Pergolide  
D1 Receptor
D2 Receptor
      98.59%
Olanzapine-d3      
D3 Receptor
    99.78%
Amisulpride-d5      
D3 Receptor
    98.27%
Adoprazine    
D2 Receptor, pA2: 9.3
D2 Receptor, pKi: 8.4
D3 Receptor, pA2: 8.9
D3 Receptor, pKi: 8.4
D4 Receptor, pKi: 8.0
  98.60%
D5R agonist 1          
D5 Receptor, EC50: 269.7 nM
99.83%
L 741742    
Human D2 Receptor, Ki: >1500 nM
Human D3 Receptor, Ki: 770 nM
Human D4 Receptor, Ki: 3.5 nM
 
L-Stepholidine  
D1 Receptor
D2 Receptor
      99.41%
Asimilobine
Dopamine Receptor
          99.9%
(Rac)-PF-06256142  
Human D1 Receptor, EC50: 107 nM
        99.59%
Bromopride    
D2 Receptor
      99.53%
Clozapine hydrochloride    
D2 Receptor, Ki: 75 nM
      99.83%
PAOPA    
D2 Receptor
      98.09%
PF-06256142  
Human D1 Receptor, EC50: 33 nM
        99.90%
Aramisulpride    
D2 Receptor, Ki: 140 nM
D3 Receptor, Ki: 13.9 nM
    98.49%
Thioridazine-d3 hydrochloride      
D3 Receptor
    98.25%
Aripiprazole monohydrate    
D2 Receptor
D3 Receptor
D4 Receptor
  99.83%
CP 226269        
D4 Receptor
  99.65%
Cariprazine-d8      
D3 Receptor
    98.77%
(-)-GSK598809 hydrochloride      
D3 Receptor
    99.64%
Brexpiprazole S-oxide-d8    
D2 Receptor, Ki: 0.3 nM
      98.72%
A-381393      
D3 Receptor
D4 Receptor
  99.92%
Ro 10-5824 dihydrochloride        
D4 Receptor
  99.86%
Perospirone hydrochloride  
D1 Receptor, Ki: 41 nM
D2 Receptor, Ki: 1.4 nM
      99.94%
Pramipexole-d5 dihydrochloride    
D2 Receptor
D3 Receptor
D4 Receptor
 
Cyclo(glycyl-L-leucyl)
Dopamine Receptor
          99.75%
Carmoxirole hydrochloride    
D2 Receptor
      99.82%
A-77636 hydrochloride    
D2 Receptor
      ≥98.0%
ABT-724 trihydrochloride        
D4 Receptor
  99.05%
Esamisulpride    
D2 Receptor
D3 Receptor
    99.04%
SKF 83959 hydrobromide  
D1 Receptor, Ki: 1.18 nM
D2 Receptor, Ki: 920 nM
D3 Receptor, Ki: 399 nM
 
D5 Receptor, Ki: 7.56 nM
99.86%
Pardoprunox hydrochloride    
D2 Receptor, pEC50: 8
D3 Receptor, pEC50: 9.2
    99.46%
Ecopipam hydrobromide  
D1 Receptor, Ki: 1.2 nM
D2 Receptor, Ki: 980 nM
 
D4 Receptor, Ki: 5520 nM
D5 Receptor, Ki: 2.0 nM
99.0%
(Rac)-Levomepromazine-d3 hydrochloride      
D3 Receptor
   
Metoclopramide hydrochloride    
D2 Receptor, IC50: 483 nM
      99.96%
Mesdopetam      
D3 Receptor
   
Risperidone-d4    
D2 Receptor
      99.34%
PD 168568 dihydrochloride    
D2 Receptor, Ki: 1842 nM
D3 Receptor, Ki: 2682 nM
D4 Receptor, Ki: 8.8 nM
  99.71%
SKF-83566 hydrobromide  
D1 Receptor
     
D5 Receptor
Zuclopenthixol dihydrochloride    
D2 Receptor
      99.98%
MLS6357      
Dopamine D3 receptor, IC50: 13 μM
    99.57%
Iloperidone carboxylic acid  
Human D1 Receptor, pKi: 5.94
 
Rat D3 Receptor, pKi: 6.11
    99.6%
Haloperidol-d4    
D2 Receptor
     
FAUC 213    
hD2 Receptor, Ki: 3.4 μM
hD3 Receptor, Ki: 5.3 μM
hD4.4 Receptor, Ki: 2.2 nM
  99.86%
S-14506 hydrochloride    
D2 Receptor
      98.64%
NGD94-1        
hD4.2 Receptor, Ki: 3.6 nM
  99.73%
Quinelorane dihydrochloride    
D2 Receptor
D3 Receptor
    99.0%
U-99194 maleate      
D3 Receptor, Ki: 160 nM
    99.23%
Mesulergine hydrochloride
Dopamine Receptor
         
DETQ  
Human D1 Receptor, EC50: 5.8 nM
       
Razpipadon  
D1 Receptor
        99.95%
MLS1082  
D1 Receptor
        99.55%
Fananserin        
D4 Receptor, Ki: 2.93 nM
  99.97%
Benzquinamide hydrochloride    
D2 Receptor
D3 Receptor
D4 Receptor
  99.14%
D3/5-HT receptor modulator-1  
D1 Receptor, Ki: 3290 nM
D2 Receptor, Ki: 263 nM
D3 Receptor, Ki: 4.5 nM
    99.75%
SKF-75670 hydrobromide  
D1 Receptor
        99.83%
(-)-Isocorypalmine  
D1 Receptor
D2 Receptor
D3 Receptor
D4 Receptor
D5 Receptor
99.67%
Mosapramine    
D2 Receptor
      98.58%
Spiramide  
D1 Receptor, Ki: 2530 nM
D2 Receptor, Ki: 3 nM
      99.23%
Clomipramine-d3 hydrochloride      
D3 Receptor
    99.98%
cis-(Z)-Flupentixol dihydrochloride    
D2 Receptor, Ki: 0.38 nM
     
Brexpiprazole S-oxide    
D2 Receptor, Ki: 0.3 nM
     
SB-277011 dihydrochloride      
D3 Receptor
   
ST-836 hydrochloride    
D2 Receptor, Ki: 132 nM
D3 Receptor, Ki: 4.5 nM
   
Risperidone hydrochloride    
D2 Receptor, Ki: 5.9 nM
     
(Rac)-Rotigotine hydrochloride  
D1 Receptor, Ki: 83 nM
D2 Receptor, Ki: 13.5 nM
D3 Receptor, Ki: 0.71 nM
D4 Receptor, Ki: 3.9-15 nM
D5 Receptor, Ki: 5.4 nM
98.11%
Moperone    
D2 Receptor, IC50: 1 nM
D3 Receptor, IC50: 1 nM
    99.5%
Aplindore    
D2 Receptor, pKi: 9.1
      98.44%
5-HT6/7 antagonist 1    
D2 Receptor
     
Zuclopenthixol-d4 succinate    
D2 Receptor
      99.0%
Risperidone-d6    
D2 Receptor, Ki: 5.9 nM
     
Ziprasidone mesylate trihydrate    
Rat D2 Receptor, Ki: 4.8 nM
     
Clocapramine    
D2 Receptor
     
Levosulpiride-d3      
D3 Receptor
    99.79%
Propionylpromazine-d6 hydrochloride    
D2 Receptor
      99.78%
Blonanserin dihydrochloride  
D1 Receptor, Ki: 1070 nM
D2 Receptor, Ki: 0.142 nM
D3 Receptor, Ki: 0.494 nM
D4 Receptor, Ki: 150 nM
 
Tetrabenazine mesylate    
D2 Receptor, Ki: ~2.1 μM
     
Amisulpride-d5 N-Oxide      
D3 Receptor
   
Paliperidone-d4    
D2 Receptor
     
Iloperidone-d3      
D3 Receptor
    98.8%
Nomifensine-d3 maleate      
D3 Receptor
   
Cabergoline-d5    
D2 Receptor
D3 Receptor
   
D1/D5 Receptor agonist-1  
D1 Receptor
     
D5 Receptor
PD 172760        
D4 Receptor
 
YM-50001        
D4 Receptor, Ki: 5.62 nM
 
Dopamine D3 receptor ligand-3    
D2 Receptor, Ki: 353 nM
D3 Receptor, Ki: 3.6 nM
   
AL-LAD  
D1 Receptor
D2 Receptor
     
PNU-177864 hydrochloride      
D3 Receptor
   
S18327    
D2 Receptor
     
PD 158771    
hD2 Receptor, Ki: 42 nM
Human D3 Receptor, Ki: 13.7 nM
   
NGD 94-1 dimaleate        
hD4.2 Receptor, Ki: 3.6 nM
 
Pramipexole-d7 dihydrochloride    
D2 Receptor
D3 Receptor
D4 Receptor
 
SK609 hydrochloride      
Dopamine D3 receptor, EC50: 1109 nM
    99.83%
Dopamine D3 receptor ligand-1    
D2 Receptor, Ki: 715 nM
D3 Receptor, Ki: 8 nM
   
D-520    
D2 Receptor, EC50: 4.73 nM
D2L Receptor, Ki: 41.8 nM
D3 Receptor, EC50: 2.18 nM
D3 Receptor, Ki: 0.35 nM
   
ARN25657      
D3 Receptor, EC50: 15.2 nM
D3 Receptor, Ki: 1.5 nM
   
5-HT1AR/5-HT6R ligand-1    
D2 Receptor, Ki: 1903 nM
     
Tropapride    
D2 Receptor
     
Piribedil dihydrochloride    
D2 Receptor
D3 Receptor
   
A68930  
D1 Receptor
       
5-HT1AR agonist 2    
D2 Receptor, Ki: 23 nM
     
BP 897    
D2 Receptor
D3 Receptor
   
UNC10062  
D1 Receptor
       
Norzine dimalate    
D2 Receptor
     
Tau-aggregation-IN-1    
D2 Receptor
D3 Receptor
   
D4R antagonist-2        
D4 Receptor
 
PNU-96415E        
D4 Receptor
 
Clomipramine-d3      
D3 Receptor
   
L 741742 hydrochloride    
Human D2 Receptor, Ki: >1500 nM
Human D3 Receptor, Ki: 770 nM
Human D4 Receptor, Ki: 3.5 nM
 
Nooglutil    
D2 Receptor
     
Melperone hydrochloride    
Human D2 Receptor, Kd: 180 nM
     
L-745870 trihydrochloride    
D2 Receptor, Ki: 960 nM
D3 Receptor, Ki: 2300 nM
Human D4 Receptor, Ki: 4.3 nM
 
5-OH-DPAT    
D2 Receptor
     
Aramisulpride hydrochloride    
D2 Receptor, Ki: 140 nM
D3 Receptor, Ki: 13.9 nM
   
PZ-1657    
D2 Receptor, Ki: 1004 nM
     
Trepipam  
D1 Receptor
       
PZ-1657 hydrochloride    
D2 Receptor, Ki: 1004 nM
     
Brexpiprazole hydrochloride    
D2L Receptor, Ki: 0.3 nM
     
Tiapride    
D2 Receptor, IC50: 110-320 nM
D3 Receptor, IC50: 180 nM
   
(S)-SKF-77434  
D1 Receptor, IC50: 2800 nM
       
CNV-dopamine    
D2 Receptor
     
SV 156    
Human D2 Receptor, Ki: 2.5 ± 0.4 nM
Human D3 Receptor, Ki: 96.9 ± 4.3 nM
Human D4 Receptor, Ki: 700 ± 56 nM
 
(S)-Remoxipride  
D1 Receptor, IC50: >100 μM
D2 Receptor, IC50: 1.57 μM
     
BP 897 hydrochloride    
D2 Receptor
D3 Receptor
    99.84%
FAUC 346      
D3 Receptor, EC50: 1.5 nM
    99.90%
AVE-5997      
D3 Receptor
   
Lirexapride    
Dopamine D2 receptor
     
N-Methylspiroperidol    
D2 Receptor
     
(Z)-Flupenthixol decanoate  
D1 Receptor
D2 Receptor
     
Dihydrexidine  
D1 Receptor, IC50: 10 nM
       
Carmoxirole    
D2 Receptor
     
5-HT2A receptor agonist-13    
D2 Receptor, Ki: 1298 nM
     
Blonanserin-d8    
D2 Receptor
     
SCH-23390 maleate  
D1 Receptor, Ki: 0.2 nM
     
D5 Receptor, Ki: 0.3 nM
(-)-GSK598809      
D3 Receptor
   
Bromocriptine-13C,d3    
D2 Receptor
D3 Receptor
   
CYD-1-79      
D3 Receptor
   
FMJ-01-054    
Human D2 Receptor, Ki: >100,000 nM
Human D3 Receptor, Ki: >100,000 nM
Human D4 Receptor, Ki: 77.7 nM
 
Promazine    
D2 Receptor
     
Raclopride tartrate  
D1 Receptor, Ki: 18000 nM
D2 Receptor, Ki: 1.8 nM
D3 Receptor, Ki: 3.5 nM
D4 Receptor, Ki: 2400 nM
 
BMS-570520    
D2 Receptor, IC50: 0.64 μM
     
Dopamine D3 receptor ligand-4    
D2 Receptor, Ki: 7.43 nM
D3 Receptor, Ki: 0.5 nM
   
Tipepidine citrate    
D2 Receptor
     
UNC9815  
D1 Receptor
       
PD 119819
Dopamine Receptor
         
Benztropine-13C,d3 mesylate    
D2 Receptor
D3 Receptor
   
Mazapertine    
D2 Receptor, Ki: <3 nM
D3 Receptor, Ki: <3 nM
D4 Receptor, Ki: <3 nM
 
Cinitapride monotartrate    
D2 Receptor
     
Ro 10-5824        
Dopamine D4 receptor
 
Metopimazine acid-d6 (hydrochloride)    
D2 Receptor
     
Dopamine D3 receptor antagonist-3      
Dopamine D3 receptor, Kd: 0.49 μM
   
Bifeprunox    
D2 Receptor, pKi: 8.83 (striatum)
     
Berupipam  
D1 Receptor
       
Alizapride-13C,d3 hydrochloride      
D3 Receptor
   
Bromopride hydrochloride    
D2 Receptor
     
Piribedil hydrochloride    
D2 Receptor
D3 Receptor
   
NRA-0562  
Human D1 Receptor, Ki: 7.09 nM
Human D2 Receptor, Ki: 2.49 nM
Human D3 Receptor, Ki: 3.48 nM
Human D4 Receptor, Ki: 1.79 nM
 
SUN-1334H free base      
Dopamine D3 receptor, IC50: 3.43 μM
   
Ordopidine    
D2 Receptor
     
EF-7412    
Dopamine D2 receptor, Ki: 22 nM
     
VK4-116      
D3 Receptor, Ki: 6.84 nM
   
Dopamine D3 receptor antagonist-1      
D3 Receptor
   
PD 118717    
D2 Receptor
     
BMY 28674    
D2 Receptor, IC50: 3.1 μM
D3 Receptor, IC50: 4.9 μM
D4 Receptor, IC50: 0.85 μM
 
Dehydrate haloperidol    
Human D2 Receptor, pKd: 8
Human D2 Receptor, pKi: 8
     
PDE1-IN-12  
D1 Receptor
       
SKF-83566-PEG1-pomalidomide  
D1 Receptor
       
Asenapine citrate  
D1 Receptor, pKi: 8.9
D2 Receptor, pKi: 8.9
D3 Receptor, pKi: 9.4
D4 Receptor, pKi: 9.0
 
Flupentixol  
D1 Receptor
D2 Receptor
     
Dopamine D2 receptor agonist-3    
D2 Receptor, EC50: 5 nM
D3 Receptor, EC50: >3.2 μM
    98.30%
SB-773812    
D2 Receptor, pKi: 7.4
D3 Receptor, pKi: 8.5
   
CSP-2503    
Dopamine D2 receptor, Ki: 192.1 nM
     
Obuprazine      
D3 Receptor, IC50: 0.37 nM
   
D1R antagonist 2  
D1 Receptor, IC50: 35.6 ( cAM nM
D1 Receptor, IC50: 70 (β-arre nM
       
Dopamine D4 receptor ligand 2    
D2 Receptor, IC50: >1000 nM
 
D4 Receptor, IC50: 0.057 nM
 
Dopamine D3 receptor antagonist-2      
D3 Receptor, Ki: 2.16 nM
   
PD-143188    
D2 Receptor, Ki: 25.5 nM
D3 Receptor, Ki: 16.6 nM
hD4.2 Receptor, Ki: 90.9 nM
 
Bromperidol hydrochloride    
D2 Receptor
      99.96%
PZ-1129    
D2 Receptor, Ki: 24 nM
     
Loxapine hydrochloride  
Human D1 Receptor
Human D2 Receptor
 
Human D4 Receptor
 
Sibenadet    
D2 Receptor
     
SSR-181507 hydrochloride    
D2 Receptor
     
SB-414796    
D2 Receptor, Ki: 400 nM
D3 Receptor, Ki: 4 nM
   
Asenapine-13C,d3 hydrochloride      
D3 Receptor
D4 Receptor
 
Dopamine D3 receptor agonist 1      
D3 Receptor, Ki: 0.268 nM
   
NGB 2904 hydrochloride      
D3 Receptor, Ki: 1.4
   
Roxindole    
D2 Receptor
     
U-99194      
D3 Receptor
   
Flupenthixol decanoate    
D2 Receptor
     
Dopamine D3 receptor ligand-2    
D2 Receptor, Ki: 1228 nM
D3 Receptor, Ki: 11.4 nM
   
Clocapramine dihydrochloride hydrate    
D2 Receptor
     
Agroclavine  
D1 Receptor
       
BGC20-761    
Human D2 Receptor, Ki: 140 nM
     
Dopamine D3 receptor agonist-2  
D1 Receptor, Ki: 4700 nM
dopamine D2L receptor, Ki: 7.67 nM
D3 Receptor, Ki: 0.268 nM
D4 Receptor, Ki: 284 nM
 
PF-4363467    
D2 Receptor, Ki: 692 nM
D3 Receptor, Ki: 3.1 nM
   
D4R antagonis-2        
D4 Receptor, IC50: 6.87 μM
 
(-)-IHCH7041    
D2 Receptor, Ki: 22.44 nM
     
Adrogolide  
D1 Receptor
       
SKF 38393 hydrobromide  
D1 Receptor, IC50: 110 nM
       
Clozapine dihydrochloride    
D2 Receptor, Ki: 75 nM
     
RU-24213 hydrochloride    
Dopamine D2 receptor
     
Itopride    
D2 Receptor
     
Haloperidol-13C6    
D2 Receptor
     
Antipsychotic agent-2    
D2 Receptor, Kb: 45.7 nM
     
PD 168568    
D2 Receptor, Ki: 1842 nM
D3 Receptor, Ki: 2682 nM
D4 Receptor, Ki: 8.8 nM
 
PF-04363467      
D3 Receptor
   
Molindone hydrochloride (Standard)    
D2 Receptor
   
D5 Receptor
UCSF34    
D2L Receptor, pKi: 7.49
     
Ziprasidone mesylate    
Rat D2 Receptor, Ki: 4.8 nM
     
NEO 376
Dopamine Receptor
          99.23%
D3R ligand 1      
D3 Receptor, Ki: 66 nM
   
A-77636  
Dopamine D1 receptor, EC50: 1.1 nM
Dopamine D1 receptor, Ki: 39.8 nM
       
A-69024  
D1 Receptor, Ki: 12.6 nM
D2 Receptor, Ki: 1290 nM
     
Perphenazine dihydrochloride    
D2 Receptor, Ki: 0.56 nM
D3 Receptor, Ki: 0.43 nM
D4 Receptor, Ki: 28.5 nM
 
Cabergoline-d6    
D2 Receptor
D3 Receptor
   
5-HT7R antagonist 3    
D2 Receptor, Ki: 511 nM
     
D2R/D3R/5-HT1AR agonist 1    
D2 Receptor, EC50: 1.29 nM
D3 Receptor, EC50: 1.05 nM
   
(Rac)-Rotigotine-d7 hydrochloride  
D1 Receptor
 
D3 Receptor
D4 Receptor
 
Acetophenazine    
D2 Receptor
      98.05%
SKF 38393  
D1 Receptor
       
7-Hydroxy-DPAT      
D3 Receptor
   
OS-3-106      
D3 Receptor, Ki: 0.2 nM
   
SKF83822 hydrobromide  
D1 Receptor
       
FGH31        
Dopamine D4 receptor, Ki: 1.6 nM
 
Dopamine D2 receptor antagonist-3    
D2 Receptor, pIC50: 5.52
     
L-750667 triHydrochloride        
D4 Receptor, Ki: 0.51 nM
D4 Receptor, Kd: 0.16 nM
  99.39%
1192U90    
D2 Receptor
     
Haloperidol-d4-1    
D2 Receptor
      98.0%
MOR agonist-2      
D3 Receptor
   
BRL 34778    
D2 Receptor, Ki: 2.14 nM
     
D4R antagonist-1        
D4 Receptor, IC50: 6.87 μM
 
Piquindone    
D2 Receptor
     
Dopamine D3 receptor ligand-6      
D3 Receptor
   
Itopride-d6 hydrochloride    
D2 Receptor
     
FLA-797  
D1 Receptor
D2 Receptor
     
Fluphenazine decanoate dihydrochloride    
D2 Receptor
     
SEP-4199    
D2 Receptor, Ki: 16 nM
     
Thioridazine 2-Sulfone-d3      
D3 Receptor
   
ABT-724        
D4 Receptor
D5 Receptor
98.04%
Risperidone mesylate    
D2 Receptor, Ki: 5.9 nM
     
Blonanserin-d5    
D2 Receptor
     
Ropinirole-d4 hydrochloride    
D2 Receptor
D3 Receptor
D4 Receptor
 
Pimozide-d5 N-Oxide  
D1 Receptor
 
D3 Receptor
   
Metopimazine-d6    
D2 Receptor
     
Melperone (Standard)    
Human D2 Receptor, Kd: 180 nM
     
Melperone-d4 hydrochloride    
Human D2 Receptor, Kd: 180 nM
      99.84%
Iloperidone hydrochloride  
Rat D1 Receptor, Ki: 546 nM
Human D1 Receptor, Ki: 216 nM
Rat D2 Receptor, Ki: 54 nM
Human D3 Receptor, Ki: 7.1 nM
Human D4 Receptor, Ki: 25 nM
Human D5 Receptor, Ki: 319 nM
(S)-SKF 38393  
D1 Receptor
       
Haloperidol-d4 N-Oxide    
D2 Receptor
     
Sumanirole    
D2 Receptor
     
ADX-10061  
D1 Receptor, Ki: 5.8 nM
D2 Receptor, Ki: > >10 000 nM
     
BRD5814    
D2 Receptor
     
FAUC-312  
Dopamine D1 receptor, Ki: 29000 nM
Dopamine D2 receptor, Ki: 25000 nM
Dopamine D3 receptor, Ki: 13000 nM
Dopamine D4 receptor, Ki: 1.5 nM
 
Pardoprunox    
D2 Receptor, pEC50: 8
D3 Receptor, pEC50: 9.2
   
Sarizotan dihydrochloride      
Human D3 Receptor, IC50: 6.8 nM
   
Dopamine D3 receptor ligand-5  
D1 Receptor, Ki: 4600 nM
D2 Receptor, Ki: 2.85 nM
D3 Receptor, Ki: 0.14 nM
D4 Receptor, Ki: 756 nM
 
Raclopride-d5 hydrochloride      
D3 Receptor
    99.82%
7-Hydroxy-PIPAT      
D3 Receptor, Ki: 0.99 nM
   
Abaperidone    
D2 Receptor, IC50: 17 nM
     
NRA-0160      
D3 Receptor, Ki: 39 nM
D4 Receptor, Ki: 0.48 nM
 
ABT-670        
D4 Receptor
 
(S)-Remoxipride hydrochloride hydrate  
D1 Receptor, IC50: >100 μM
D2 Receptor, IC50: 1.57 μM
     
SNAP8719 free base    
D2 Receptor, pKi: 5.98
     
Desethoxy Quetiapine dihydrochloride    
D2 Receptor, IC50: 1330 nM
     
SKF 83509    
D2 Receptor, Ki: 70.2 nM
     
Cariprazine impurity 1    
D2 Receptor
     
BL-1020 mesylate    
D2S Receptor, Ki: 0.062 nM
D2L Receptor, Ki: 0.066 nM
     
FR 64822    
D2 Receptor
     
Lurasidone metabolite 14326    
D2 Receptor
     
U-101958 maleate    
D2 Receptor, IC50: 1980 nM
D3 Receptor, IC50: 552 nM
D4 Receptor, IC50: 2.7 nM
 
Benzquinamide    
D2 Receptor
D3 Receptor
D4 Receptor